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Long-Term Use of Ticagrelor in Patients with Prior Myocardial Infarctionopen access

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Bonaca, Marc P.Bhatt, Deepak L.Cohen, MarcSteg, Philippe GabrielStorey, Robert F.Jensen, Eva C.Magnani, GiuliaBansilal, SameerFish, M. PollyIm, KyungahBengtsson, OlofOphuis, Ton OudeBudaj, AndrzejTheroux, PierreRuda, MikhailHamm, ChristianGoto, ShinyaSpinar, JindrichNicolau, Jose CarlosKiss, Robert G.Murphy, Sabina A.Wiviott, Stephen D.Held, PeterBraunwald, EugeneSabatine, Marc S.PEGASUS-TIMI 54 Steering Committee and InvestigatorsMorin, SuzanneFish, M. PollyDantzer, EmilyAcquilano, DayleMcGuire, Rachael L.Gannon, Joseph B.Gershman, ElaineIm, KyungAhAhlbom, Ann MaxeBoberg, BarbroAbola, Maria TeresaArdissino, DiegoAylward, PhilipBudaj, AndrzejCorbalan, RamonDalby, AnthonyDellborg, MikaelDiaz, RafaelDimulescu, DoinaGoto, ShinyaGoudev, AssenGuneri, SemaHamm, ChristianHu, DayiIsaza, DanielKamensky, GabrielKiss, RobertKontny, FredericLopez-Sendon, JoseMedina, FelixMontalescot, GillesNicolau, JosePaolasso, ErnestoParkhomenko, AlexanderRuda, MikhailSeung, Ki-BaeVan de Werf, FransAnderson, Jeffrey L.White, Harvey D.Verheugt, Freek W. A.Pedersen, Terje R.DeMets, David L.Lowe, CherylArevalo, ChristinaAwtry, EricBerger, CliffordCroce, KevinDesai, AkshayGelfand, EliHo, CarolynLeeman, DavidLink, MarkNorden, AndrewPande, AshvinRost, NataliaRuberg, FrederickSilverman, ScottSinghal, AneeshVita, JosephAlvarisqueta, A.De Gennaro, N.Berli, M.Roude, A. E.Di Gennaro, J. AlbisuAlbisu, J. F.Caccavo, A.Torres, M.Cuadrado, J.Bordoni, P.Cuello, J.Aviles, A.Glenny, A.Recoaro, R.Fernandez, R.Strada, B. N.Fuentealba, V.Gallo, C.Duran, R. Garc-aGarcia, C.Hominal, M.Castoldi, M.Jure, H.Pacora, F. FerreLorenzatti, A.Martinez, J. M.Macin, S.Cocco, N.MacKinnon, I.Bagnato, M. B.Marino, J.Cusimano, S.Arias, V.Focaccia, M.Muntaner, J.Mansilla, V.Poy, C.Prado, A.Paterlini, G.Montana, O.Camino, A.Sala, J.Luciani, C.Vico, M.Morell, Y.Dumont, C.Vottero, E.Zangroniz, P.Lescano, A.Morara, P.Marquez, L. LoboPatron, F. RissoLabarta, G. BustamanteSivila, C. D.Quiroga, A. R.Maffei, L.Sassone, S.Rolandi, F.Vesentini, N.Carnero, G.Del Verme, S.Hershson, A.Figal, J. C.Viso, M. E.Hii, C.Smith, K.Singh, B.Acampo, M.Rogers, J.ODonoghue, M.Amerena, J.Long, A.Dart, A.Kay, S.Worthley, M.Nimmo, J.Lehman, R.Morrison, H.Dick, R.Savage, C.van Gaal, W.Park, M.Blombery, P.McCarthy, C.Oqueli, E.Hill, D.Sader, M.Vrachas, D.Purnell, P.Vibert, J.Collins, N.Gordon, A.Arstall, M.Rose, J.Aroney, C.Cleave, P.Fitzpatrick, M.Mackenzie, M.Garrahy, P.Hall, C.Nelson, G.Reid, E.Lee, A.Gibbs, J.Thompson, P.Crittenden, J.Hammett, C.Hindom, L.Antonis, P.Manzoney, A.Cross, D.Pollard, C.Brieger, D.Wu, J.Whelan, A.Tulloch, G.Taylor, A.Smith, B.Horowitz, J.Black, M.Boland, J.Malmendier, D.Celen, H.Wendelen, E.Claeys, M.Pieter, M.Cools, F.Simons, N.De Maeseneire, S.De Wolf, L.Brike, C.Dubois, P.Bolado, A. Conde Y.Foading-Deffo, B.Tahon, S.Friart, A.Arend, C.Gevaert, S.Verdegem, P.Marechal, P.Gits, F.Pierard, L.Celentano, C.Pirenne, B.Bouvy, C.Renkin, J.Huyberechts, D.Sinnaeve, P.De Velder, L.Stammen, F.Casier, T.Striekwold, H.Van den Broeck, D.Thoeng, J.Goris, R.Timmermans, P.Collard, S. -J.van de Borne, P.De Clippel, M.Wollaert, B.Jacobs, C.Vankelecom, B.Daelemans, Y.Vervoort, G.Drieghe, S.Vranckx, P.Janssen, A.Vrolix, M.I., SimenonWijns, W.Delacroix, H.Denie, D.Schoors, D.Lemoine, I.Cornelis, K.Willems, A. -M.Schroder, E.Domange, J.Greque, G.Machado, H.Armaganijan, D.Del Monaco, M. I.da Silva, D.Nakazone, R.Dutra, O.R., VazDaher, R.Rodrigues, D.Guimaraes, A.Teixeira, A.Saraiva, J.Costa, M.Leaes, P.Blacher, M.Maia, L.Nakazone, MA.Manenti, E.Ruschel, K.Marin-Neto, J.Pavao, R.Preto, RiberaoJunior, A. AlvesOliveira, G.Rassi, S.Sampaio, D.Rossi, P. R.dos Santos, L.de Souza, J.Lino, E.Pimentel Filho, P.Zucchetti, C.Gomes, M.de Paiva, A.Sousa, A. C.Almeida, A.Botelho, R.da Silva, R.Giraldez, R.Franken, M.Faludi, A.Bertolami, M.Hernandes, M.Lucas, N.Carvalho, A.Bertolami, A.Precoma, D.Geralde, L.Pereira, A.Cesar, L.Mioto, B.Marino, R.Rabelo, W.dos Santos, F.Vidotti, M. 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Issue Date
May-2015
Publisher
Massachusetts Medical Society
Citation
New England Journal of Medicine, v.372, no.19, pp 1791 - 1800
Pages
10
Indexed
SCI
SCIE
SCOPUS
Journal Title
New England Journal of Medicine
Volume
372
Number
19
Start Page
1791
End Page
1800
URI
https://scholarworks.korea.ac.kr/kumedicine/handle/2020.sw.kumedicine/7887
DOI
10.1056/NEJMoa1500857
ISSN
0028-4793
1533-4406
Abstract
BACKGROUND The potential benefit of dual antiplatelet therapy beyond 1 year after a myocardial infarction has not been established. We investigated the efficacy and safety of ticagrelor, a P2Y12 receptor antagonist with established efficacy after an acute coronary syndrome, in this context. METHODS We randomly assigned, in a double-blind 1:1:1 fashion, 21,162 patients who had had a myocardial infarction 1 to 3 years earlier to ticagrelor at a dose of 90 mg twice daily, ticagrelor at a dose of 60 mg twice daily, or placebo. All the patients were to receive low-dose aspirin and were followed for a median of 33 months. The primary efficacy end point was the composite of cardiovascular death, myocardial infarction, or stroke. The primary safety end point was Thrombolysis in Myocardial Infarction (TIMI) major bleeding. RESULTS The two ticagrelor doses each reduced, as compared with placebo, the rate of the primary efficacy end point, with Kaplan–Meier rates at 3 years of 7.85% in the group that received 90 mg of ticagrelor twice daily, 7.77% in the group that received 60 mg of ticagrelor twice daily, and 9.04% in the placebo group (hazard ratio for 90 mg of ticagrelor vs. placebo, 0.85; 95% confidence interval [CI], 0.75 to 0.96; P=0.008; hazard ratio for 60 mg of ticagrelor vs. placebo, 0.84; 95% CI, 0.74 to 0.95; P=0.004). Rates of TIMI major bleeding were higher with ticagrelor (2.60% with 90 mg and 2.30% with 60 mg) than with placebo (1.06%) (P<0.001 for each dose vs. placebo); the rates of intracranial hemorrhage or fatal bleeding in the three groups were 0.63%, 0.71%, and 0.60%, respectively. CONCLUSIONS In patients with a myocardial infarction more than 1 year previously, treatment with ticagrelor significantly reduced the risk of cardiovascular death, myocardial infarction, or stroke and increased the risk of major bleeding. (Funded by AstraZeneca; PEGASUS-TIMI 54 ClinicalTrials.gov number, NCT01225562. opens in new tab.)
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Anam Hospital (Department of Cardiology, Anam Hospital)
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